AZ PFKFB3 26

CAS No. 1704740-52-2

AZ PFKFB3 26( —— )

Catalog No. M26619 CAS No. 1704740-52-2

AZ PFKFB3 26 is an effective and selective PFKFB3 inhibitor with an IC50 of 23 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 40 Get Quote
5MG 65 Get Quote
10MG 115 Get Quote
25MG 260 Get Quote
50MG 447 Get Quote
100MG 624 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    AZ PFKFB3 26
  • Note
    Research use only, not for human use.
  • Brief Description
    AZ PFKFB3 26 is an effective and selective PFKFB3 inhibitor with an IC50 of 23 nM.
  • Description
    AZ PFKFB3 26 is an effective and selective PFKFB3 inhibitor with an IC50 of 23 nM. The IC50s for PFKFB1 and PFKFB2 are 2.06 and 0.384 μM, respectively.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    Glucokinase
  • Recptor
    Human Endogenous Metabolite
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1704740-52-2
  • Formula Weight
    402.498
  • Molecular Formula
    C24H26N4O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 5 mg/mL (12.42 mM)
  • SMILES
    CC(C)Cn1cc(C#N)c2cc(Oc3ccc(NC(=O)[C@@H]4CCCN4)cc3)ccc12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Biratsi A, et al. A highly conserved mechanism for the detoxification and assimilation of the toxic phytoproduct L-azetidine-2-carboxylic acid in Aspergillus nidulans. Sci Rep. 2021 Apr 1;11(1):7391.
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